Back to Single Peptide Protocols
Single PeptideMetabolic & Weight Loss20 mg vialWeeklySubcutaneousGLP-1/GIP/Glucagon

Retatrutide (20 mg Vial) Dosage Protocol

Full dosage protocol for the triple-agonist GLP-1/GIP/glucagon receptor peptide in a 20 mg vial. Includes titration schedule.

Vial Size
20 mg
Route
Subcutaneous
Frequency
Once weekly
Dose Range
2–12 mg/week

Dosage Schedule

PeriodDose
Weeks 1–42 mg
Weeks 5–84 mg
Weeks 9–128 mg
Weeks 13+12 mg

Route: Subcutaneous · Frequency: Once weekly · Cycle: 24–52 weeks

How It Works

Retatrutide is a triple-receptor agonist targeting GLP-1, GIP, and glucagon receptors simultaneously. Phase 2 trials showed 24.2% body weight reduction at 48 weeks — the highest reported for any weekly injectable.

Potential Benefits

  • Phase 2: 24.2% mean weight loss at 48 weeks (highest of any weekly injectable).
  • Triple mechanism: appetite suppression + energy expenditure + fat oxidation.
  • Significant improvement in metabolic markers.

Side Effects & Risks

  • Nausea, vomiting, diarrhea (dose-dependent).
  • Currently in Phase 3 trials; not yet FDA-approved.

Important Notes

  • Investigational compound — not FDA-approved.
  • Titrate slowly to minimize GI side effects.

Storage Instructions

  • Lyophilized: −20 °C (−4 °F).
  • Once mixed: 2–8 °C; use within 28 days.

References

  1. [1]Jastreboff AM et al. Triple-Hormone-Receptor Agonist Retatrutide for Obesity. NEJM 2023.View Source

Research & Educational Use Only: This protocol is for educational and research purposes only. It does not constitute medical advice, diagnosis, or treatment. Always consult a qualified healthcare professional before making any decisions related to peptides or any other compounds.